A. A. Zubenko, A. S. Morkovnik, L. N. Divaeva, O. P. Demidov, V. S. Sochnev, I. G. Borodkina, Yu. D. Drobin, A. A. Spasov, “New route to bioactive 2-(hetero)arylethylamines <i>via</i> nucleophilic ring opening in fused 7-acyl-2,3-dihydroazepines”, Mendeleev Commun., 2020, Volume 30, Issue 1,Pages <nobr>28–30</nobr>

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Mendeleev Commun., 2020 Volume 30, Issue 1, Pages 28–30 (Mi mendc1090)

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Communications

New route to bioactive 2-(hetero)arylethylamines via nucleophilic ring opening in fused 7-acyl-2,3-dihydroazepines

A. A. Zubenko^a, A. S. Morkovnik^b, L. N. Divaeva^b, O. P. Demidov^c, V. S. Sochnev^b, I. G. Borodkina^b, Yu. D. Drobin^a, A. A. Spasov^d

^a North-Caucasian Zonal Research Veterinary Institute, Novocherkassk, Russian Federation
^b Institute of Physical and Organic Chemistry, Southern Federal University, Rostov-on-Don, Russian Federation
^c North-Caucasus Federal University, Stavropol, Russian Federation
^d Volgograd State Medical University, Volgograd, Russian Federation

Abstract: Nucleophilic heterocyclic ring opening in fused 7-acyl- H+ 1,2-dihydroazepines with o-phenylenediamine affords b-(hetero)arylethylamines.

Keywords: fused dihydroazepines, azepine–pyrazine recyclization, baryl(heteroaryl)ethylamines, bioactive amines, ring opening reactions.

Language: English

DOI: 10.1016/j.mencom.2020.01.009

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