E. S. Matyugina, A. L. Khandazhinskaya, S. N. Kochetkov, K. L. Seley-Radtke, “Synthesis of 3-hetarylpyrroles by Suzuki–Miyaura cross-coupling”, Mendeleev Commun., 2020, Volume 30, Issue 2,Pages <nobr>231

This article is cited in 10 papers

Communications

Synthesis of 3-hetarylpyrroles by Suzuki–Miyaura cross-coupling

E. S. Matyugina^a, A. L. Khandazhinskaya^a, S. N. Kochetkov^a, K. L. Seley-Radtke^b

^a V.A. Engelhardt Institute of Molecular Biology, Russian Academy of Sciences, Moscow, Russian Federation
^b Department of Chemistry and Biochemistry, University of Maryland, Maryland, USA

Abstract: 1-[tert-Butyl(diphenyl)silyl]pyrrol-3-ylboronic acid was obtained from pyrrole in three steps. Its Suzuki–Miyaura cross-coupling with functionalized pyridinyl and pyrimidinyl bromides afforded new promising 3-hetaryl-1H-pyrroles.

Keywords: heterocyclic aromatic compounds, fleximers, Suzuki–Miyaura cross-coupling, pyrrole, iodination, silyl protection.

Language: English

DOI: 10.1016/j.mencom.2020.03.034

	*Supplementary materials:*
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