A. N. Vereshchagin, M. N. Elinson, A. D. Korshunov, M. P. Egorov, “Highly efficient one-pot cascade cyclization of 3-(5-hydroxy-3-methylpyrazol-4-yl)-3-arylpropionitriles into spirocyclopropyl pyrazolones”, Mendeleev Commun., 2016, Volume 26, Issue 1,Pages <nobr>19

This article is cited in 4 papers

Communications

Highly efficient one-pot cascade cyclization of 3-(5-hydroxy-3-methylpyrazol-4-yl)-3-arylpropionitriles into spirocyclopropyl pyrazolones

A. N. Vereshchagin, M. N. Elinson, A. D. Korshunov, M. P. Egorov

N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Moscow, Russian Federation

Abstract: Bromine-assisted one-pot cascade cyclization of 3-(5-hydroxy-3-methylpyrazol-4-yl)-3-arylpropionitriles affords medicinally relevant spirocyclopropyl pyrazolones in 60–97% yields.

Language: English

DOI: 10.1016/j.mencom.2016.01.008

	*Supplementary materials:*
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